张荣, 钱旭红, 宋伟荣, 庄建治. N-(5-芳基-1,3,4-噁二唑-2-基)-取代酰胺的合成及生物活性[J]. 农药学学报, 1999, 1(2): 88-90.
    引用本文: 张荣, 钱旭红, 宋伟荣, 庄建治. N-(5-芳基-1,3,4-噁二唑-2-基)-取代酰胺的合成及生物活性[J]. 农药学学报, 1999, 1(2): 88-90.
    Zhang Rong, Qian Xu-hong, Song Wei-rong, Zhuang Jian-zhi. SYNTHESIS AND BIOACTIVITY OF N(5ARYL 1,3,4OXADIAZOL2YL)SUBSTITUTED AMIDES[J]. Chinese Journal of Pesticide Science, 1999, 1(2): 88-90.
    Citation: Zhang Rong, Qian Xu-hong, Song Wei-rong, Zhuang Jian-zhi. SYNTHESIS AND BIOACTIVITY OF N(5ARYL 1,3,4OXADIAZOL2YL)SUBSTITUTED AMIDES[J]. Chinese Journal of Pesticide Science, 1999, 1(2): 88-90.

    N-(5-芳基-1,3,4-噁二唑-2-基)-取代酰胺的合成及生物活性

    SYNTHESIS AND BIOACTIVITY OF N(5ARYL 1,3,4OXADIAZOL2YL)SUBSTITUTED AMIDES

    • Abstract: Acylation of 2-amio-5-aryl-1,3,4-oxadiazoles with acyl chlorides and trichloroacetic acid to afford eleven new -N--5-aryl-1,3,4-oxadiazol-2-yl-substituted amides. The required oxadiazole precursors are prepared by oxidative cyclization of corresponding aldehyde semicarbazones. The structures of the synthesized compounds are elucidated by elemental analysis、 1HNMR、IR and MS. They are screened for their larvicidal activities against wild fruit and antibiotic activities.

       

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