岳敏, 袁勤坤, 金林红. 含酰腙结构的新型吡唑酰胺衍生物对小菜蛾的生物活性[J]. 农药学学报, 2012, 14(4): 449-452.
    引用本文: 岳敏, 袁勤坤, 金林红. 含酰腙结构的新型吡唑酰胺衍生物对小菜蛾的生物活性[J]. 农药学学报, 2012, 14(4): 449-452.
    YUE Min, YUAN Qinkun, JIN Linhong. Insecticidal activities of novel pyrazole amides containing hydrazone substructures against Plutella xylostella[J]. Chinese Journal of Pesticide Science, 2012, 14(4): 449-452.
    Citation: YUE Min, YUAN Qinkun, JIN Linhong. Insecticidal activities of novel pyrazole amides containing hydrazone substructures against Plutella xylostella[J]. Chinese Journal of Pesticide Science, 2012, 14(4): 449-452.

    含酰腙结构的新型吡唑酰胺衍生物对小菜蛾的生物活性

    Insecticidal activities of novel pyrazole amides containing hydrazone substructures against Plutella xylostella

    • 摘要: 采用浸虫法、夹毒叶片法和叶碟法分别测定了13个含酰腙结构的新型吡唑酰胺衍生物对小菜蛾3龄幼虫的触杀、胃毒和拒食活性。结果表明:该类化合物对小菜蛾3龄幼虫具有较高的胃毒和拒食活性,其中苯环上含有氯原子、且酰腙一端的取代基含有杂原子且体积较小的化合物 H7的胃毒和拒食活性最好,明显高于对照药剂毒死蜱。H7 72 h胃毒作用LC50值为0.6 mg/L(毒死蜱的LC50值为7.4 mg/L);有10个化合物的拒食活性高于毒死蜱,其中 H7 48 h的拒食中浓度(AFC50) 最低,为0.6 mg/L,明显低于毒死蜱(AFC50=6.5 mg/L)。供试化合物对小菜蛾3龄幼虫均无触杀活性。

       

      Abstract: Thirteen novel pyrazole amides containing hydrazine moiety were detected for their contact,stomach and anti-feeding activity in laboratory against the 3rd instar larvae of Plutella xylostella ,by using insect-dipping method,leaf sandwich method and leaf disc method respectively.The results showed that these compounds possessed high stomach activity and anti-feeding activity against the larvae.Among these compounds, H7 ,which contains chlorine atoms in benzene ring and heteroatom in the acylhydrazone moiety,had the strongest contact and stomach activity which is much higher than that of control agent chlorpyrifos.The results indicated that the LC50 value of 72 h stomach toxicity of H7 and chlorpyrifos against P. xylostella were 0.6 and 7.4 mg/L,respectively.Additionally,there were 10 compounds that showed higher anti-feeding activity than that of chlorpyrifos against P. xylostella ,and the 48 h AFC50 (concentration causing 50% antifeedant rate) value of H7 was 0.6 mg/L, while that of chlorpyrifos was 6.5 mg/L.All tested compounds showed no contact activity against P.xylostella.

       

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